Boron-trihalide-promoted regioselective ring-opening reactions of gem-difluorocyclopropyl ketones.

نویسندگان

  • Tang-Po Yang
  • Qiang Li
  • Jin-Hong Lin
  • Ji-Chang Xiao
چکیده

Boron trihalide-promoted ring-opening reactions of gem-difluorocyclopropyl ketones to give the corresponding β-trifluoromethyl ketones and β-halodifluoromethyl ketones were described. It was found that boron trihalides act as both Lewis acids and nucleophiles and the proximal bond prefers to cleave in this transformation.

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عنوان ژورنال:
  • Chemical communications

دوره 50 9  شماره 

صفحات  -

تاریخ انتشار 2014